Diseases 2 associated indications
Drugs 0 with a known mechanism
Trials 0 via those drugs
Companies 0 on linked trials

Structure

AlphaFold model for P43246 · mean pLDDT 85.3

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Identity

Synonyms, protein accessions, and subcellular locations

Synonyms

COCA1 DNA mismatch repair protein Msh2 DNA mismatch repair protein Msh2 transcript FCC1 HNPCC HNPCC1 LCFS2 LYNCH1 MMRCS2 MSH-2 MSH2 MutS protein homolog 2 MutS-like 2 hMSH2 mutS homolog 2, colon cancer, nonpolyposis type 1

Protein IDs

ensembl_PRO ENSP00000233146 ensembl_PRO ENSP00000384199 ensembl_PRO ENSP00000442697 ensembl_PRO ENSP00000495455 ensembl_PRO ENSP00000495543 ensembl_PRO ENSP00000495641 ensembl_PRO ENSP00000496351 ensembl_PRO ENSP00000496441 ensembl_PRO ENSP00000519159 ensembl_PRO ENSP00000519165 ensembl_PRO ENSP00000519166 ensembl_PRO ENSP00000519172 ensembl_PRO ENSP00000519219 ensembl_PRO ENSP00000580467 ensembl_PRO ENSP00000580468 ensembl_PRO ENSP00000588159 ensembl_PRO ENSP00000588160 ensembl_PRO ENSP00000588161 ensembl_PRO ENSP00000588162 ensembl_PRO ENSP00000588163 ensembl_PRO ENSP00000588164 ensembl_PRO ENSP00000588165 ensembl_PRO ENSP00000588166 ensembl_PRO ENSP00000588167 ensembl_PRO ENSP00000616875 uniprot_obsolete B4E2Z2 uniprot_obsolete O75488 uniprot_swissprot P43246 uniprot_trembl A0A2R8Y6P0 uniprot_trembl A0A2R8Y713 uniprot_trembl A0A2R8Y7S8 uniprot_trembl A0A2R8YFH0 uniprot_trembl A0A2R8YG02 uniprot_trembl A0AAQ5BH31 uniprot_trembl A0AAQ5BH33 uniprot_trembl A0AAQ5BH41 uniprot_trembl A0AAQ5BH48 uniprot_trembl A0AAQ5BH55 uniprot_trembl E9PHA6

Subcellular location

Cellular component Nucleoplasm

Pipeline by phase

Trial momentum

Associated diseases

2 indications loaded

Disease Score Best evidence Drugged here?
ovarian cancer
MONDO_0008170
0.74
Genetic literature No
non-small cell lung carcinoma
MONDO_0005233
0.43
Literature No

Evidence mix

What the association scores rest on

Evidence type Associations Best score
Literature 2 0.721
Somatic mutation 2 0.767
Genetic association 1 0.861
Genetic literature 1 0.865
RNA expression 1 0.104

Literature concepts

What papers discuss for this target

Mechanism of action

Cytotoxic 158 Inhibitor 134 Immune checkpoint blockade 83 Kinase inhibition 14 Immunomodulation 5

Modality

Small molecule 12 Oligonucleotide 11 Antibody 9 Cell therapy 5 CAR-T 4

Payload

Topoisomerase I inhibitor 18 DXd 16 Maytansinoid 14 DM1 11 SN-38 6

Linker

Cleavable 21 GGFG tetrapeptide 16 Non-cleavable 11 SMCC 11 mc-vc-PAB 7

Technology

CRISPR 7 Single-cell sequencing 2

Therapy area

Oncology 743 Pathological conditions 317 Urology / nephrology 270 Endocrinology 244 Gastroenterology / hepatology 200

Baseline expression

Highest nTPM by tissue, cell type, and cell line

Tissue

TissuenTPM
retina32.4
thymus30.4
tonsil23.4
lymph node22.3
testis15.2
bone marrow15.0
thyroid gland15.0
breast14.8
rectum14.1
parathyroid gland13.9
cerebral cortex13.3
cerebellum13.3

Cell type

Cell typenTPM
cone photoreceptor cells294.0
rod photoreceptor cells158.9
erythrocyte progenitors145.5
early primary spermatocytes117.5
brain inhibitory neurons113.6
distal convoluted tubule cells109.4
brain excitatory neurons97.1
differentiating spermatogonia94.9
megakaryocyte-erythroid progenitors87.4
renal connecting tubule cells84.3
pituitary stem cells83.2
retinal bipolar cells83.0

Cell line

Cell linenTPM
TK [Human B-cell lymphoma]211.6
MFM-223163.0
JM-1146.6
NTERA-2146.1
BL-70127.7
U-698-M127.4
DMS 79127.3
Farage122.8
NCI-H187121.4
SU-DHL-8119.7
EB3 [Human Burkitt lymphoma]118.2
SU-DHL-5118.1